Publications

Berti F., Frecer V., Miertuš S.: Inhibitors of HIV-protease from computational design. A history of theory and synthesis still to be fully appreciated. Curr. Pharm. Des. 20(21), 3398-3411 (2014).

Bialopiotrowicz T., Janczuk B., Fiedorowicz, Khachtryan G., Tomasik P., Bakoš D.: Hyaluronan-lecitin foils and their properties, Mater. Chem. Phys. 95, 99-104 (2006).

Bonini C, Chiummiento L, Di Blasio N, Funicello M, Lupattelli P, Tramutola F, Berti F, Ostric A, Miertuš S, Frecer V, Kong DX.: Synthesis and biological evaluation of new simple indolic non peptidic HIV Protease inhibitors: the effect of different substitution patterns. Bioorg. Med. Chem. 22(17), 4792-802 (2014).

Bubeníková, S., Lacík, I., Bakoš, D., Vodná, L.: Chitosan polyelectrolyte comlexes for use in tissue engineering and drug delivery, J. Mat. Sci. 539-543, 577-582 (2007).

Dali, B., Keita, M., Megnassan, E., Frecer, V., Miertuš, S.: Insight into selectivity of peptidomimetic inhibitors with modified statine core for plasmepsin II of Plasmodium falciparum over human cathepsin D. Chem. Biol. Drug Des. 79(4), 411-430 (2012).

Hajzer, V., Fišera, R., Latika, A., Durmis, J., Kollár, J., Frecer, V., Tučeková, Z., Miertuš, S., Kostolanský, F., Varečková, E., Šebesta, R.: Stereoisomers of oseltamivir - synthesis, in silico prediction and biological evaluation. Org. Biomol. Chem. 15(8), 1828-1841 (2017).

Harvanová D., Rosocha J., Bakoš D., Švihla R., Vaško G., Horňák S., Ledecký V., Gromošová S., Cibur P., Raši R., Collagen/hyaluronan membrane as a scaffold for chondrocytes cultivation, Biologia 64(5), 1032-1038 (2009).

Kollar J., Frecer, V.: Selective inhibitors of zinc-dependent histone deacetylases. Therapeutic targets relevant to cancer. Curr. Pharm. Des. 21(11), 1472-1502 (2015).

Kongkamnerd J, Cappelletti L, Prandi A, Seneci P, Rungrotmongkol T, Jongaroonngamsang N, Rojsitthisak P, Frecer V, Milani A, Cattoli G, Terregino C, Capua I, Beneduce L, Gallotta A, Pengo P, Fassina G, Miertus S, De-Eknamkul W.: Synthesis and in vitro study of novel neuraminidase inhibitors against avian influenza virus. Bioorg. Med. Chem. 20(6), 2152-7 (2012).

Kouassi AF, Kone M, Keita M, Esmel A, Megnassan E, N'Guessan YT, Frecer V, Miertuš S.: Computer-aided design of orally bioavailable pyrrolidine carboxamide inhibitors of enoyl-acyl carrier protein reductase of Mycobacterium tuberculosis with favorable pharmacokinetic profiles. Int. J. Mol. Sci. 16(12), 29744-29771 (2015).

Kukolikova L, Bakos D, Alexy P, et al.: Optimization of the properties of chitosan lactate/hyaluronan film, J. Appl. Polymer Sci. 100 (2), 1413-1419 (2006).

Megnassan E, Keita M, Bieri C, Esmel A, Frecer V, Miertus S.: Design of novel dihydroxynaphthoic acid inhibitors of Plasmodium falciparum lactate dehydrogenase. Med. Chem. 8(5), 970-84 (2012).

Owono Owono LC, Keita M, Megnassan E, Frecer V, Miertus S.: Design of Thymidine Analogues Targeting Thymidilate Kinase of Mycobacterium tuberculosis. Tuberc. Res. Treat. 2013(e670836), (2013).

Palou, M., Bakoš, D., Kuzielová, E., Labuda, J.: Potential Application of Glass and Glass-Ceramics Based on Lithium Disilicate as Biomaterials, Key Engineering Materials, 361-363, 273-276 (2008).

Poruban D., Bakoš D., Danišovič L., Bohmer D., Blaško M., Vojtaššak J.: In vitro prepared autologous graft from bucal mucosa - clinical application, Case Rep. Clin. Pract. Rev. 6, 62-67 (2005).

Svetlik, J., Pronayova, N., Frecer, V., Ciez, D.: Three-component reaction and organocatalysis in one: synthesis of densely substituted 4-aminochromanes. Tetrahedron 72(47), 7620-7627 (2016).

Šimon P., Chaudhry Q., Bakoš D.: Migration of engineered nanoparticles from polymer packaging to food - a physicochemical view, J. Food Nutr. Res. 47(3), 105-113 (2008).

Šimon, P., Zhong, W., Bakoš, D., Hynek, D.: Thermooxidative stability of polymethyl methacrylate containing nanoparticles of silica/titania and silica/zirconia, Chem. Pap. 62(2), 176-180 (2008).

Toti, K. S., Verbeke, F., Risseeuw, M. D. P., Frecer, V., Munier-Lehmann, H., Van Calenbergh, S.: Synthesis and evaluation of 5'-modified thymidines and 5-hydroxymethyl-2'-deoxyuridines as M. tuberculosis thymidylate kinase inhibitors. Bioorgan. Med. Chem. 21(1), 257-268 (2013).

Udommaneethanakit T, Rungrotmongkol T, Frecer V, Seneci P, Miertus S, Bren U.: Drugs against avian influenza a virus: design of novel sulfonate inhibitors of neuraminidase N1. Curr. Pharm. Des. 20(21), 3478-87 (2014).

Vittekova M., Dragunova J., Kabat P., Bozikova M., Bakos D., Koller J.: Cytotoxicity testing of scaffolds potentially suitable for the preparation of three-dimensional skin substitutes, Cell Tissue Bank. 15(3), 345-55 (2014).

Vodná, L., Bubeníková, S., Bakoš, D.: Chitosan based hydrogel microspheres as drug carriers, Macromol. Biosci. 7, 629-634 (2007).